MW 256.79 g/mol, Purity >99%. α₂ Adrenoceptor agonist (IC₅₀ = 68.2 nM). Ki values for receptor subtypes are 1570 (α₂A), 1360 (α₂B), 1200 (α₂C) and 1460 nM (α₂D). Activates KATP channels through the NO/cGMP pathway. Displays anaesthetic, antinociceptive and muscle relaxatory actions.
The product is subject to the following: Abcam Restricted Use Statement